Name: CAS: 1346574-57-9 | GSK126, NX21682
Brand: Apollo Scientific
SKU: NX21682-1MG
Price: 203.0 USD
Availability: InStock

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Product Identifiers

Catalog #	NX21682
CAS Number	1346574-57-9
PubChem CID	68210102
Chemical Name	GSK126
IUPAC Name	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methyl-6-(6-piperazin-1-ylpyridin-3-yl)indole-4-carboxamide
Synonym	EZH2 Inhibitor, GSK-2816126-A
InChI	InChI=1S/C31H38N6O2/c1-6-22(5)37-18-20(3)29-25(30(38)34-17-26-19(2)13-21(4)35-31(26)39)14-24(15-27(29)37)23-7-8-28(33-16-23)36-11-9-32-10-12-36/h7-8,13-16,18,22,32H,6,9-12,17H2,1-5H3,(H,34,38)(H,35,39)/t22-/m0/s1
InChIKey	FKSFKBQGSFSOSM-QFIPXVFZSA-N
SMILES	CC[C@H](C)n1cc(C)c2c(cc(cc12)c3ccc(nc3)N4CCNCC4)C(=O)NCc5c(C)cc(C)nc5O
MDL Number	MFCD23381067

Specification

MW	526.7
MF	C31H38N6O2
Product Notes	GSK126 is a potent, highly selective EZH2 methyltransferase inhibitor with IC50 of 9.9 nM, > 1000-fold selective for EZH2 over 20 other human methyltransferases.
Cat Number	BISN0124
Manufacturer	Apollo Scientific
Country of Origin	United Kingdom

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