CAS: 1652591-81-5 | GSK484, >98%, NX27786

SKU: NX27786-5MG
CAS: 1652591-81-5 | GSK484, >98%, NX27786
CAS: 1652591-81-5 | GSK484, >98%, NX27786

CAS: 1652591-81-5 | GSK484, >98%, NX27786

SKU: NX27786-5MG
Pack Size
Regular price $350.00
Only 0 items in stock!
  • Scholar Citation
  • SSL-Secure Payments
  • UN Approved Packaging
  • Worldwide Express Delivery

Product Identifiers

Catalog # NX27786
CAS Number 1652591-81-5
PubChem CID 86340151
Chemical Name GSK484
IUPAC Name [(3S,4R)-3-amino-4-hydroxypiperidin-1-yl]-[2-[1-(cyclopropylmethyl)indol-2-yl]-7-methoxy-1-methylbenzimidazol-5-yl]methanone;hydrochloride
Synonym PAD4 inhibitor
InChI InChI=1S/C27H31N5O3.ClH/c1-30-25-20(11-18(13-24(25)35-2)27(34)31-10-9-23(33)19(28)15-31)29-26(30)22-12-17-5-3-4-6-21(17)32(22)14-16-7-8-16;/h3-6,11-13,16,19,23,33H,7-10,14-15,28H2,1-2H3;1H/t19-,23+;/m0./s1
SMILES Cl.COc1cc(cc2nc(c3cc4ccccc4n3CC5CC5)n(C)c12)C(=O)N6CC[C@@H](O)[C@@H](N)C6
MDL Number MFCD30343874


MW 510
MF C27H32ClN5O3
Assay >98%
Product Notes GSK484 is a reversible and selective inhibitor of PAD4 with IC50 of 50 nM. GSK484 blocks the citrullination of PAD4 target proteins in human neutrophils and inhibits the formation of neutrophil extracellular traps in both mouse and human neutrophils.
Cat Number BISN0052
Manufacturer Apollo Scientific
Country of Origin United Kingdom

Request MSDS & CoA

This site is protected by reCAPTCHA and the Google Privacy Policy and Terms of Service apply.

Recently viewed